{"id":1467,"date":"2017-08-17T06:49:42","date_gmt":"2017-08-17T06:49:42","guid":{"rendered":"https:\/\/nolvadex-pct.info\/historie-nolvadexu\/"},"modified":"2017-08-17T06:49:42","modified_gmt":"2017-08-17T06:49:42","slug":"historie-nolvadexu","status":"publish","type":"page","link":"https:\/\/nolvadex-pct.info\/cs\/historie-nolvadexu\/","title":{"rendered":"Historie Nolvadexu"},"content":{"rendered":"<h2>O p\u0159\u00edpravku Nolvadex<\/h2>\n<hr>\n<p>Stejn\u011b jako u ka\u017ed\u00e9ho produktu, se kter\u00fdm se setk\u00e1te v anabolick\u00e9m v\u00fdklenku (jak\u00fdkoli produkt, kter\u00fd je ofici\u00e1ln\u011b od farmaceutick\u00e9 spole\u010dnosti dod\u00e1vaj\u00edc\u00ed polo\u017eky t\u00e9to povahy do l\u00e9ka\u0159sk\u00e9 oblasti p\u0159inejmen\u0161\u00edm), tato polo\u017eka za\u010dala \u017eivot jako prost\u0159edek k l\u00e9\u010db\u011b nemoci.<\/p>\n<p>Nebyl to v\u0161ak v\u017edy snadn\u00fd \u017eivot &#8211; tamoxifen (v\u011bdeck\u00fd n\u00e1zev pro nolvadex) vznikl v 50. letech minul\u00e9ho stolet\u00ed na z\u00e1klad\u011b \u0159ady v\u00fdzkumn\u00fdch operac\u00ed, jejich\u017e c\u00edlem bylo objevit n\u011bjakou \u00fa\u010dinnou l\u00e9\u010dbu po antikoncep\u010dn\u00ed pilulce (co\u017e se samoz\u0159ejm\u011b nakonec poda\u0159ilo).<\/p>\n<p>Tamoxifen byl poprv\u00e9 syntetizov\u00e1n a\u017e v roce 1966 (to znamen\u00e1, \u017ee se na n\u011bm pracovalo 16 let) &#8211; a\u010dkoli se neuk\u00e1zal b\u00fdt p\u0159\u00edli\u0161 \u00fa\u010dinn\u00fd jako antikoncep\u010dn\u00ed prost\u0159edek, <strong>slibn\u011b p\u016fsobil jako l\u00e9k proti rakovin\u011b<\/strong>.<\/p>\n<p>Navzdory tomuto p\u0159\u00edslibu FDA ud\u011blila patent na tuto slou\u010deninu a\u017e v 80. letech 20. stolet\u00ed (na po\u010d\u00e1tku) a pr\u00e1v\u011b zde jsme poprv\u00e9 vid\u011bli nolvadex jako formu l\u00e9\u010dby rakoviny v prvn\u00ed linii. M\u016f\u017eeme dodat, \u017ee s velk\u00fdm \u00fa\u010dinkem. <\/p>\n<p>Jakmile si kulturistick\u00e1 komunita uv\u011bdomila, \u017ee m\u016f\u017ee \u00fa\u010dinn\u011b kontrolovat hladinu estrogenu (kulturist\u00e9 t\u00e9 doby m\u011bli pouze z\u00e1kladn\u00ed biologick\u00e9 znalosti o chemii steroid\u016f, ale bylo pom\u011brn\u011b v\u0161eobecn\u011b zn\u00e1mo, \u017ee estrogen hraje velkou roli v ne\u017e\u00e1douc\u00edch slo\u017ek\u00e1ch u\u017e\u00edv\u00e1n\u00ed steroid\u016f), za\u010dalo se experimentovat a nolvadex je od t\u00e9 doby <a href=\"https:\/\/nolvadex-pct.info\/cs\/proc-pouzivat-nolvadex-behem-pct\/\">v\u00fdznamnou sou\u010d\u00e1st\u00ed kulturistick\u00fdch cykl\u016f<\/a>.<\/p>\n<p>Je t\u0159eba poznamenat, \u017ee tamoxifen byl pou\u017e\u00edv\u00e1n v obdob\u00ed p\u0159ed 80. lety v d\u016fsledku toho, \u017ee se n\u011bkter\u00fdm jedinc\u016fm dostaly do rukou experiment\u00e1ln\u00ed varianty t\u00e9to l\u00e1tky ur\u010den\u00e9 pouze pro v\u00fdzkumn\u00e9 \u00fa\u010dely.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"aligncenter size-full wp-image-300\" src=\"https:\/\/nolvadex-pct.info\/wp-content\/uploads\/2018\/08\/history-of-nolvagen-main.jpg\" alt=\"\" width=\"650\" height=\"300\"><\/p>\n<h2>L\u00e9ka\u0159sk\u00e9 pou\u017eit\u00ed Nolvadex<\/h2>\n<hr>\n<p class=\"Normal1\" style=\"text-align: justify;\"><span lang=\"EN\" style=\"font-size: 14.0pt; line-height: 115%;\">Obvykle uvid\u00edte, \u017ee nolvadex se pou\u017e\u00edv\u00e1 v r\u00e1mci l\u00e9ka\u0159sk\u00e9 kapacity pro n\u00e1sleduj\u00edc\u00ed \u00fa\u010dely:<\/span><\/p>\n<ul id=\"mycheck\">\n<li>Rakovina prsu<\/li>\n<li>Neplodnost<\/li>\n<li>Gynekomastie<\/li>\n<\/ul>\n<p>Pokud jde o posledn\u00ed polo\u017eku na seznamu, nolvadex se uk\u00e1zal b\u00fdt obzvl\u00e1\u0161t\u011b \u00fa\u010dinn\u00fd proti vzniku gynekomastie vzhledem k tomu, \u017ee se zam\u011b\u0159uje na p\u016fsoben\u00ed sv\u00fdch \u00fa\u010dink\u016f v prsn\u00ed tk\u00e1ni t\u011bla.<\/p>\n<p>Je to vzhledem k tomu, \u017ee estrogen projev na tomto konkr\u00e9tn\u00edm m\u00edst\u011b je to, co vede ke gynekomastie, \u017ee nolvadex se uk\u00e1\u017ee b\u00fdt tak brut\u00e1ln\u011b \u00fa\u010dinn\u00fd v t\u00e9to kapacit\u011b.<\/p>\n<p>P\u0159i sledov\u00e1n\u00ed jeho \u00fa\u010dinnosti jako pomocn\u00edka p\u0159i neplodnosti je pom\u011brn\u011b snadn\u00e9 pochopit, jak a pro\u010d se pro tento \u00fa\u010del osv\u011bd\u010duje. Nolvadex (stejn\u011b jako v\u0161echny p\u0159\u00edpravky SERM) ve skute\u010dnosti slou\u017e\u00ed ke zv\u00fd\u0161en\u00ed produkce LH i FSH. Respektive tyto hormony jsou v pln\u00e9m zn\u011bn\u00ed zn\u00e1my jako <a href=\"http:\/\/www.vivo.colostate.edu\/hbooks\/pathphys\/endocrine\/hypopit\/lhfsh.html\" target=\"_blank\" rel=\"nofollow noopener\">luteiniza\u010dn\u00ed hormon a folikuly stimuluj\u00edc\u00ed hormon<\/a>.  <\/p>\n<p><strong>Oba tyto hormony jsou \u017eivotn\u011b d\u016fle\u017eit\u00e9 pro produkci testosteronu<\/strong>, proto jak\u00e9koli zv\u00fd\u0161en\u00ed jejich p\u0159\u00edtomnosti okam\u017eit\u011b znamen\u00e1, \u017ee hladina testosteronu se zv\u00fd\u0161\u00ed.<\/p>\n<p>Pokud jde o l\u00e9\u010dbu rakoviny prsu &#8211; stejn\u00fd mechanismus \u00fa\u010dinku, kter\u00fd vede k regresi gynekomastie, vede tak\u00e9 k regresi rakoviny prsu.<\/p>\n<p>Bylo prok\u00e1z\u00e1no, \u017ee rakovinn\u00e9 bu\u0148ky (zejm\u00e9na ty, kter\u00e9 se pod\u00edlej\u00ed na vzniku rakoviny prsu) se v prsn\u00ed tk\u00e1ni \u017eiv\u00ed estrogenem. Pou\u017eit\u00edm nolvadexu sni\u017eujeme obsah estrogenu p\u0159\u00edmo v t\u00e9to oblasti, co\u017e znamen\u00e1, \u017ee od\u0159\u00edzneme zdroj paliva pro rakovinu. <\/p>\n<h2>Schv\u00e1lila Sv\u011btov\u00e1 zdravotnick\u00e1 organizace<\/h2>\n<hr>\n<p class=\"Normal1\" style=\"text-align: justify;\"><span lang=\"EN\" style=\"font-size: 14.0pt; line-height: 115%;\">Nolvadex je <\/span><span lang=\"EN\"><a href=\"http:\/\/www.who.int\/medicines\/publications\/essentialmedicines\/18th_EML.pdf\" target=\"_blank\" rel=\"nofollow noopener\"><span style=\"font-size: 14.0pt; line-height: 115%; color: #1155cc;\">schv\u00e1len pro l\u00e9\u010dbu<\/span><\/a><\/span><span lang=\"EN\" style=\"font-size: 14.0pt; line-height: 115%;\"> Sv\u011btovou zdravotnickou organizac\u00ed a je uveden na seznamu \u00fa\u010dinn\u00fdch l\u00e9k\u016f pro uveden\u00e9 \u00fa\u010dely.<\/span><\/p>\n<p class=\"Normal1\" style=\"text-align: justify;\"><span lang=\"EN\" style=\"font-size: 14.0pt; line-height: 115%;\"> <\/span><span lang=\"EN\" style=\"font-size: 14.0pt; line-height: 115%;\">Toto potvrzen\u00ed znamen\u00e1, \u017ee m\u016f\u017eete m\u00edt jistotu, \u017ee pou\u017e\u00edv\u00e1te n\u011bco, co je vyzkou\u0161en\u00e9 a testovan\u00e9 a co je pova\u017eov\u00e1no za schopn\u00e9 p\u0159in\u00e9st m\u011b\u0159iteln\u00fd a v\u00fdznamn\u00fd rozd\u00edl p\u0159i pou\u017eit\u00ed ve v\u00fd\u0161e uveden\u00fdch sc\u00e9n\u00e1\u0159\u00edch.<\/span><\/p>\n<h2>Pro\u010d tedy pou\u017e\u00edvat Nolvadex?<\/h2>\n<hr>\n<p class=\"Normal1\" style=\"text-align: justify;\">Je to opr\u00e1vn\u011bn\u00e1 ot\u00e1zka &#8211; poj\u010fme nyn\u00ed sledovat mechaniku, pro\u010d a jak opravdu mus\u00edte za\u010d\u00edt br\u00e1t nolvadex v\u00e1\u017en\u011b (a v\u0161echny ostatn\u00ed formy ochrany), pokud se chyst\u00e1te pou\u017e\u00edvat anabolick\u00e9 steroidy.<\/p>\n<h3>\u00da\u010dinky zv\u00fd\u0161en\u00e9 hladiny estrogenu na t\u011blo<\/h3>\n<p>Lid\u00e9 si obvykle spojuj\u00ed zv\u00fd\u0161enou hladinu estrogenu s estetick\u00fdm po\u0161kozen\u00edm, ale ve skute\u010dnosti mohou b\u00fdt \u00fa\u010dinky mnohem hlub\u0161\u00ed a mohou v\u00e9st k trval\u00e9mu du\u0161evn\u00edmu a fyzick\u00e9mu po\u0161kozen\u00ed.<\/p>\n<p>Vysok\u00e1 m\u00edra zadr\u017eov\u00e1n\u00ed vody m\u00e1 nap\u0159\u00edklad negativn\u00ed vliv na definici sval\u016f, ale hlavn\u011b vede k potenci\u00e1ln\u011b zv\u00fd\u0161en\u00e9mu krevn\u00edmu tlaku v d\u016fsledku stla\u010dov\u00e1n\u00ed c\u00e9vn\u00edch st\u011bn.<\/p>\n<p>Gynekomastie tak\u00e9 vypad\u00e1 nevzhledn\u011b, ale ve skute\u010dnosti je to v\u00e1\u017en\u011bj\u0161\u00ed stav, ne\u017e si lid\u00e9 uv\u011bdomuj\u00ed. Kdy\u017e se gynekomastie rozvine do ur\u010dit\u00e9ho stupn\u011b, je nejen nevratn\u00e1, ale m\u016f\u017ee v\u00e9st i k rozvoji rakovinn\u00fdch bun\u011bk. <\/p>\n<p>To znamen\u00e1, \u017ee to, co se mohlo zd\u00e1t jako &#8222;ne\u0161kodn\u00fd&#8220; flirt se steroidy, m\u016f\u017ee skon\u010dit nutnost\u00ed operace, pokud nebudete \u00fa\u010dinn\u011b kontrolovat hladinu estrogenu; v nejhor\u0161\u00edm p\u0159\u00edpad\u011b se u v\u00e1s vyvine \u017eivot ohro\u017euj\u00edc\u00ed onemocn\u011bn\u00ed.<\/p>\n<p>Jako by tyto probl\u00e9my nesta\u010dily, pokud by se va\u0161e endokrinn\u00ed rovnov\u00e1ha (vnit\u0159n\u00ed rovnov\u00e1ha va\u0161\u00ed hormon\u00e1ln\u00ed aktivity) vy\u0159adila ze synchronizace, pak <strong>byste mohli skon\u010dit s v\u00e1\u017en\u011b vy\u010derpanou schopnost\u00ed produkovat a vyu\u017e\u00edvat testosteron<\/strong>. Obnoven\u00ed t\u011bchto hladin p\u0159irozenou cestou bez ochrany m\u016f\u017ee trvat a\u017e rok. <\/p>\n<h3>Rychl\u00e1 normalizace po cyklu<\/h3>\n<p>D\u00edky schopnosti nolvadexu zvy\u0161ovat hladiny FSH a LH jsme nakonec schopni rychle obnovit hladiny testosteronu po anabolick\u00e9m cyklu.<\/p>\n<p><strong>Tyto \u017eivotn\u011b d\u016fle\u017eit\u00e9 hormony n\u00e1m umo\u017e\u0148uj\u00ed vytvo\u0159it siln\u00fd z\u00e1klad pro produkci testosteronu<\/strong> a omladit na\u0161i kapacitu pro jeho vnit\u0159n\u00ed ob\u011bh. Bez p\u0159\u00edpravku, jako je nolvadex, m\u016f\u017ee trvat a\u017e rok, ne\u017e se hladiny samy pln\u011b obnov\u00ed. <\/p>\n","protected":false},"excerpt":{"rendered":"<p>O p\u0159\u00edpravku Nolvadex Stejn\u011b jako u ka\u017ed\u00e9ho produktu, se kter\u00fdm se setk\u00e1te v anabolick\u00e9m v\u00fdklenku (jak\u00fdkoli produkt, kter\u00fd je ofici\u00e1ln\u011b od farmaceutick\u00e9 spole\u010dnosti dod\u00e1vaj\u00edc\u00ed polo\u017eky t\u00e9to povahy do l\u00e9ka\u0159sk\u00e9 oblasti p\u0159inejmen\u0161\u00edm), tato polo\u017eka za\u010dala \u017eivot jako prost\u0159edek k l\u00e9\u010db\u011b nemoci. Nebyl to v\u0161ak v\u017edy snadn\u00fd \u017eivot &#8211; tamoxifen (v\u011bdeck\u00fd n\u00e1zev pro nolvadex) vznikl v 50. [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"parent":0,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"","meta":{"footnotes":""},"class_list":["post-1467","page","type-page","status-publish","hentry"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v26.9 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Historie Nolvadexu | Nolvadex-PCT<\/title>\n<meta name=\"description\" content=\"Tamoxifen byl poprv\u00e9 syntetizov\u00e1n a\u017e v roce 1966.P\u0159e\u010dt\u011bte si o historii a pou\u017eit\u00ed p\u0159\u00edpravku Nolvadex a o tom, jak se stal obl\u00edben\u00fdm p\u0159\u00edpravkem kulturist\u016f.\" \/>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/nolvadex-pct.info\/cs\/historie-nolvadexu\/\" \/>\n<meta property=\"og:locale\" content=\"cs_CZ\" \/>\n<meta property=\"og:type\" 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